Increase of leishmanicidal and tubercular activities using steroids linked to aminoquinoline
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چکیده
منابع مشابه
Increase of leishmanicidal and tubercular activities using steroids linked to aminoquinoline
UNLABELLED BACKGROUND Aminoquinoline/steroid conjugates were synthesized based on the fact that steroid transporters have been shown to accept and carry a variety of drugs. So, in continuing our research of antileishmanial and antitubercular drugs, aminoquinoline/steroid conjugates (12, 13, and 14) were regioselectively synthesized via 1, 3-dipolar cycloaddition of alkynes 3, 5, and 7 with a...
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ژورنال
عنوان ژورنال: Organic and Medicinal Chemistry Letters
سال: 2012
ISSN: 2191-2858
DOI: 10.1186/2191-2858-2-16